A Phase 1/2 Study of CYT-0851 in B-Cell Malignancies and Advanced Solid Tumors

Part of paid clinical trials in San Francisco, California.

Sponsor
Cyteir Therapeutics, Inc.
Study ID
NCT03997968
Phase
PHASE1/PHASE2
Status
Completed

Conditions

Eligibility Criteria

Sex
ALL
Age
18 Years - N/A
Healthy Volunteers
Not accepted

Interventions

  • CYT-0851 — DRUG
    Part A and B: Daily oral doses of CYT-0851 for 28 day cycles
  • CYT-0851 in combination with gemcitabine — DRUG
    Part D: Daily oral doses of CYT-0851 for 28 days in combination with gemcitabine
  • CYT-0851 in combination with capecitabine — DRUG
    Part E: Daily oral doses of CYT-0851 for 21 days in combination with capecitabine
  • CYT-0851 in combination with rituximab and bendamustine — DRUG
    Part C: Daily oral doses of CYT-0851 for 28 days in combination with rituximab and bendamustine

Study Details

This clinical trial is an interventional, active-treatment, open-label, multi-center, Phase 1/2 study. The study objectives are to assess the safety, tolerability and pharmacokinetics (PK) of CYT-0851 in patients with relapsed/refractory B-cell malignancies and advanced solid tumors and to identify a recommended Phase 2 dose as a monotherapy and in combination with chemotherapy for evaluation in these patients.

Key Dates

Start date
Oct 9, 2019
Status verified
Dec 2024
Primary completion
Nov 30, 2024
Completion
Dec 20, 2024

Study Design

Enrollment
169 participants (actual)
Allocation
NON_RANDOMIZED
Intervention model
SEQUENTIAL
Primary purpose
TREATMENT

Arms

  • Experimental: CYT-0851 dose escalation
    Part A: CYT-0851 administered orally in rising doses QD or BID for 28 day cycles
  • Experimental: CYT-0851 dose expansion
    Part B: CYT-0851 administered orally at the selected Phase 2 dose for 28 day cycles
  • Experimental: CYT-0851 and rituximab and bendamustine
    Part C: Daily oral doses of CYT-0851 for 28 days in combination with rituximab on Day 1 and bendamustine on Days 1 and 2 of each 28 day cycle
  • Experimental: CYT-0851 and gemcitabine
    Part D: Daily oral doses of CYT-0851 for 28 days in combination with gemcitabine on Day 1, 8 and 15 of each 28 day cycle
  • Experimental: CYT-0851 and capecitabine
    Part E: Daily oral doses of CYT-0851 for 21 days in combination with capecitabine on Days to 14 of each 21 day cycle

Primary Outcome Measure

Part A: Incidence of dose limiting toxicity [ Time Frame: 28 Days ]

Locations (16)

FacilityCityStateZIPSite coordinators
University of California San FranciscoSan FranciscoCalifornia94158-
Stanford Comprehensive Cancer CenterStanfordCalifornia94305-
Sarah Cannon Research Institute at HealthONEDenverColorado80218-
Florida Cancer Specialists and Research InstituteSarasotaFlorida34232-
Dana Farber Cancer InstituteBostonMassachusetts02115-
Massachusetts General HospitalBostonMassachusetts02114-
University of MichiganAnn ArborMichigan48109-
Mayo ClinicRochesterMinnesota55905-
John Theurer Cancer Center at HUMCHackensackNew Jersey07601-
NYU Langone HealthNew YorkNew York10016-
Oklahoma University-Stephenson Cancer CenterOklahoma CityOklahoma73104-
Thomas Jefferson University, Sidney Kimmel Cancer CenterPhiladelphiaPennsylvania19107-
Sarah Cannon Research Institute at Tennessee OncologyNashvilleTennessee37203-
The University of Texas MD Anderson Cancer CenterHoustonTexas77030-
University of Washington Seattle Cancer CenterSeattleWashington98109-
Medical College of WisconsinMilwaukeeWisconsin53226-

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