A Study to Examine the Effects of Esomeprazole on the Pharmacokinetics of Orally Administered Lapatinib in Subjects With Metastatic ErbB2 Positive Breast Cancer

Part of paid clinical trials in Greenville, South Carolina.

Sponsor
GlaxoSmithKline
Study ID
NCT00849329
Phase
PHASE1
Status
Completed

Conditions

  • Neoplasms, Breast

Eligibility Criteria

Sex
ALL
Age
18 Years - 65 Years
Healthy Volunteers
Not accepted

Interventions

  • lapatinib — DRUG
    1250mg lapatinib
  • lapatinib plus esomeprazole — DRUG
    1250mg lapatinib plus esomeprazole 40mg

Study Details

This study will characterize the effect of elevated gastric pH mediated by the proton-pump inhibitor, esomeprazole, on the relative bioavailability of lapatinib in subjects with metastatic ErbB2 positive breast cancer.

Key Dates

Start date
Mar 10, 2009
Status verified
Nov 2017
Primary completion
Nov 24, 2009
Completion
Nov 24, 2009

Study Design

Enrollment
12 participants (actual)
Allocation
NON_RANDOMIZED
Intervention model
SINGLE_GROUP
Primary purpose
TREATMENT

Arms

  • Experimental: Period 1
    1250mg lapatinib once daily in the morning
  • Experimental: Period 2
    1250mg lapatinib once daily in the morning in combination with esomeprazole 40mg once daily at bedtime.

Primary Outcome Measure

The area under the concentration versus time curve, minimum observed concentration, maximum observed concentration, time at which it occurs, and lag time in the appearance of measurable plasma concentrations of lapatinb [ Time Frame: Continue until disease progression or withdrawal consent ]

Locations (1)

FacilityCityStateZIPSite coordinators
GSK Investigational SiteGreenvilleSouth Carolina29605-

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