A Study to Investigate the Pharmacokinetics and Safety of Remibrutinib in Participants With Hepatic Impairment Compared With Matched Healthy Participants
- Sponsor
- Novartis Pharmaceuticals
- Study ID
- NCT05753592
- Phase
- PHASE1
- Status
- Completed
Conditions
- Hepatic Impairment
Eligibility Criteria
- Sex
- ALL
- Age
- 18 Years - 70 Years
- Healthy Volunteers
- Accepted
Interventions
- Part 1; LOU064 (Remibrutinib) — DRUG25 mg remibrutinib (5.5 days)
- Part 2; LOU064 (Remibrutinib) — DRUG25 mg remibrutinib (5.5 days)
Study Details
This was a Phase 1, open-label study to evaluate the PK, safety, and tolerability after administration of multiple doses of remibrutinib in participants with mild, moderate, or severe hepatic impairment (HI) compared to pooled matched healthy control participants with normal hepatic function.
Key Dates
- Start date
- Oct 31, 2022
- Status verified
- May 2025
- Primary completion
- Dec 14, 2023
- Completion
- Dec 17, 2023
Study Design
- Enrollment
- 38 participants (actual)
- Allocation
- NON_RANDOMIZED
- Intervention model
- CROSSOVER
- Primary purpose
- TREATMENT
Arms
- Experimental: Part 1; LOU064 (Remibrutinib)Mild and Moderate HI participants and matching healthy participants
- Experimental: Part 2; LOU064 (Remibrutinib)Severe HI participants and matching healthy participants
Primary Outcome Measure
Cmax,ss [ Time Frame: 72 hours ]
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