Study of MP0533 in Patients Acute Myeloid Leukemia or Myelodysplastic Syndrome
- Sponsor
- Molecular Partners AG
- Study ID
- NCT05673057
- Phase
- PHASE1/PHASE2
- Status
- Active Not Recruiting
Conditions
- Acute
- Leukemia
- Myeloid
- Newly Diagnosed
Eligibility Criteria
- Sex
- ALL
- Age
- 18 Years - N/A
- Healthy Volunteers
- Not accepted
Interventions
- MP0533 (multispecific DARPin CD3 Engager Targeting CD33, CD123 and CD70) monotherapy, Part 1 — DRUGMP0533 is administered by intravenous infusion
- MP0533 (multispecific DARPin CD3 Engager Targeting CD33, CD123 and CD70) monotherapy, Part 2-Arm A — DRUG* MP0533 is administered by intravenous infusion * Obinutuzumab pretreatment administered
- MP0533 (multispecific DARPin CD3 Engager Targeting CD33, CD123 and CD70) + azacitidine + venetoclax — DRUG* MP0533 is administered by intravenous infusion * Azacitidine is administered by subcutaneous injection for 7 days per cycle * Venetoclax is administered orally for 14 days per cycle * Optional obinutuzumab pretreatment administered
- MP0533 with Obinutuzumab pretreatment — DRUG* MP0533 is administered by intravenous infusion at densified dosing schedule * Obinutuzumab pretreatment administered
- MP0533 + azacitidine + venetoclax with optional Obinutuzumab pretreatment, Arm B relapsed/refractory AML — DRUG* MP0533 is administered by intravenous infusion * Azacitidine is administered by subcutaneous injection for 7 days per cycle * Venetoclax is administered orally for 14 days per cycle * Optional obinutuzumab pretreatment administered
- MP0533 + azacitidine + venetoclax with optional Obinutuzumab pretreatment, Arm B in treatment naïve patients — DRUG* MP0533 is administered by intravenous infusion * Azacitidine is administered by subcutaneous injection for 7 days per cycle * Venetoclax is administered orally for 14 days per cycle * Optional obinutuzumab pretreatment administered
Study Details
The purpose of this study is to evaluate the safety, tolerability, and preliminary activity of MP0533 in patients with acute myeloid leukemia (AML) or myelodysplastic syndrome (MDS)
Key Dates
- Start date
- Dec 29, 2022
- Status verified
- Jun 2026
- Primary completion
- May 29, 2026
- Completion
- May 31, 2027
Study Design
- Enrollment
- 249 participants (estimated)
- Allocation
- NON_RANDOMIZED
- Intervention model
- SEQUENTIAL
- Primary purpose
- TREATMENT
Arms
- Experimental: Dose escalation (Part 1)• MP0533 is administered by intravenous infusion
- Experimental: Dose escalation (Part 2 - Arm A)* MP0533 is administered by intravenous infusion * Obinutuzumab pretreatment administered
- Experimental: Dose escalation (Part 2 - Arm B)* MP0533 is administered by intravenous infusion * Azacitidine is administered by subcutaneous injection for 7 days per cycle * Venetoclax is administered orally for 14 days per cycle * Optional Obinutuzumab pretreatment administered
- Experimental: Dose expansion (Arm A)* MP0533 is administered by intravenous infusion at densified dosing schedule * Obinutuzumab pretreatment administered
- Experimental: Dose expansion (Arm B relapsed/refractory AML)* MP0533 is administered by intravenous infusion * Azacitidine is administered by subcutaneous injection for 7 days per cycle * Venetoclax is administered orally for 14 days per cycle * Optional Obinutuzumab pretreatment administered
- Experimental: Dose expansion (Arm B in treatment naïve patients)* MP0533 is administered by intravenous infusion * Azacitidine is administered by subcutaneous injection for 7 days per cycle * Venetoclax is administered orally for 14 days per cycle * Optional obinutuzumab pretreatment administered
Primary Outcome Measure
Phase 1 dose escalation: Recommended Phase 2 Dose Regimen and/or Maximum Tolerated Dose Regimen [ Time Frame: from start of treatment to end of first cycle (day 1 - 28) ]
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