A Study to Assess Zibotentan Pharmacokinetics in Participants With Moderate Hepatic and Moderate Renal Impairment
- Sponsor
- AstraZeneca
- Study ID
- NCT05112419
- Phase
- PHASE1
- Status
- Completed
Conditions
- Hepatic Impairment
- Renal Impairment
Eligibility Criteria
- Sex
- ALL
- Age
- 18 Years - 80 Years
- Healthy Volunteers
- Accepted
Interventions
- Zibotentan — DRUGAll participants will receive a single oral dose of zibotentan capsule under fasted conditions.
Study Details
This study will evaluate the pharmacokinetics (PK), safety, and tolerability of a single oral dose of zibotentan in patients with moderate hepatic and moderate renal impairment in comparison to a matched healthy control group.
Key Dates
- Start date
- Nov 10, 2021
- Status verified
- Jan 2022
- Primary completion
- Dec 15, 2021
- Completion
- Dec 15, 2021
Study Design
- Enrollment
- 12 participants (actual)
- Allocation
- NON_RANDOMIZED
- Intervention model
- PARALLEL
- Primary purpose
- TREATMENT
Arms
- Experimental: Cohort 1: Participants with moderate hepatic impairment and moderate renal impairmentParticipants will receive a single oral dose of zibotentan under fasted conditions.
- Experimental: Cohort 2: Healthy participantsParticipants will receive a single oral dose of zibotentan under fasted conditions.
Primary Outcome Measure
Area under plasma concentration-time curve from time zero to infinity (AUCinf) [ Time Frame: Day 1 to Day 6 ]
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